Details for Patent: 5,912,238
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Summary for Patent: 5,912,238
Title: | Heteroatoms-containing tricyclic compounds |
Abstract: | The invention concerns the compounds of formula I ##STR1## wherein the substituents have various significances. They are prepared by several processes including epimerizing replacement, treatment with cyanogen bromide or thiophosgene, treatment with an acid having a non-nucleophilic anion, treatment with dimethylsulfoxide and acetic anhydride, acylation, treatment with an oxalyl derivative and ammonia, methylation, oxidation, deprotection and protection. They possess interesting pharmacological activity as antiinflammatory, immunosuppressant, antiproliferative and chemotherapeutic drug resistance reversing agents. |
Inventor(s): | Baumann; Karl (Vienna, AT), Emmer; Gerhard (Vienna, AT) |
Assignee: | Novartis AG (Basel, CH) |
Application Number: | 08/276,276 |
Patent Claim Types: see list of patent claims | Compound; Composition; Use; |
Drugs Protected by US Patent 5,912,238
Applicant | Tradename | Generic Name | Dosage | NDA | Approval Date | TE | Type | RLD | RS | Patent No. | Patent Expiration | Product | Substance | Delist Req. | Patented / Exclusive Use | Submissiondate |
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>Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
Foreign Priority and PCT Information for Patent: 5,912,238
International Family Members for US Patent 5,912,238
Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
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European Patent Office | 0427680 | ⤷ Sign Up | 91021 | Luxembourg | ⤷ Sign Up |
European Patent Office | 0427680 | ⤷ Sign Up | SPC/GB03/015 | United Kingdom | ⤷ Sign Up |
European Patent Office | 0427680 | ⤷ Sign Up | 300134 | Netherlands | ⤷ Sign Up |
European Patent Office | 0427680 | ⤷ Sign Up | SZ 12/2003 | Austria | ⤷ Sign Up |
European Patent Office | 0427680 | ⤷ Sign Up | 12/2003 | Austria | ⤷ Sign Up |
Austria | 126803 | ⤷ Sign Up | |||
Australia | 640963 | ⤷ Sign Up | |||
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