Details for Patent: 5,965,525
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Summary for Patent: 5,965,525
Title: | Cyclic peptide antifungal agents |
Abstract: | Provided are compounds of the formula (1): ##STR1## wherein R' is hydrogen, methyl or NH.sub.2 C(O)CH.sub.2 --; R" and R'" are independently methyl or hydrogen; R and R.sup.y are independently hydroxy or hydrogen; R.sub.1 is hydroxy, hydrogen, or hydroxysulfonyloxy; R.sub.7 is hydroxy, hydrogen, hydroxysulfonyloxy or phosphonooxy; R.sub.2 is a novel acyl side chain. Also provided are novel formulations, methods of inhibiting fungal and parasitic activity, and a process for preparing dideoxy (R=H) forms of the compounds. |
Inventor(s): | Burkhardt; Frederick J. (Indianapolis, IN), Debono; Manuel (Indianapolis, IN), Nissen; Jeffrey S. (Indianapolis, IN), Turner, Jr.; William W. (Bloomington, IN) |
Assignee: | Eli Lilly and Company (Indianapolis, IN) |
Application Number: | 08/449,056 |
Patent Claim Types: see list of patent claims | Compound; Use; Composition; Formulation; | More… ↓ |
Drugs Protected by US Patent 5,965,525
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>Applicant | >Tradename | >Generic Name | >Dosage | >NDA | >Approval Date | >TE | >Type | >RLD | >RS | >Patent No. | >Patent Expiration | >Product | >Substance | >Delist Req. | >Patented / Exclusive Use | >Submissiondate |
International Family Members for US Patent 5,965,525
Country | Patent Number | Estimated Expiration | Supplementary Protection Certificate | SPC Country | SPC Expiration |
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European Patent Office | 0561639 | ⤷ Subscribe | 91406 | Luxembourg | ⤷ Subscribe |
European Patent Office | 0561639 | ⤷ Subscribe | CA 2008 00017 | Denmark | ⤷ Subscribe |
European Patent Office | 0561639 | ⤷ Subscribe | 300334 | Netherlands | ⤷ Subscribe |
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