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Last Updated: September 26, 2024

Details for Patent: 7,511,041


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Which drugs does patent 7,511,041 protect, and when does it expire?

Patent 7,511,041 protects ALIQOPA and is included in one NDA.

This patent has fifty patent family members in thirty-two countries.

Summary for Patent: 7,511,041
Title:Fused azole-pyrimidine derivatives
Abstract: The present invention relates to hovel fused azolepyrimidine derivatives, processes for preparing them and pharmaceutical preparations containing them. The fused azolepyrimidine derivatives of the present invention exhibit enhanced potency for phosphotidylinositol-3-kinase (PI3K) inhibition, especially for PI3K-.gamma. inhibition and can be used for the prophylaxis and treatment of diseases associated with PI3K and particularly with PI3K-.gamma. activity. More specifically, the azole derivatives of the present invention are useful for treatment and prophylaxis of diseases as follows: inflammatory and immunoregulatory disorders, such as asthma, atopic dermatitis, rhinitis, allergic diseases, chronic obstructive pulmonary disease (COPD), septic shock, joint diseases, autoixnmune pathologies such as rheumatoid arthritis, and Graves' disease, cancer, myocardial contractility disorders, heart failure, thromboembolism, ischemia, and atherosclerosis. The compounds of the present invention are also useful for pulmonary hypertension, renal failure, cardiac hypertrophy, as well as neurodegenerative disorders such as Parkinson's disease, Alzheimer's disease, diabetes and focal ischemia, since the diseases also relate to PI3K activity in a human or animal subject.
Inventor(s): Shimada; Mitsuyuki (Nara, JP), Murata; Toshiki (Nara, JP), Fuchikami; Kinji (Tokyo, JP), Tsujishita; Hideki (Kyoto, JP), Omori; Naoki (Hyogo, JP), Kato; Issei (Nara, JP), Miura; Mami (Nara, JP), Urbahns; Klaus (Lund, SE), Gantner; Florian (Constance, DE), Bacon; Kevin (San Diego, CA)
Assignee: Bayer Pharmaceuticals Corporation (West Haven, CT)
Application Number:10/527,376
Patent Claim Types:
see list of patent claims
Composition; Compound;

Drugs Protected by US Patent 7,511,041

Applicant Tradename Generic Name Dosage NDA Approval Date TE Type RLD RS Patent No. Patent Expiration Product Substance Delist Req. Patented / Exclusive Use Submissiondate
Bayer Healthcare ALIQOPA copanlisib dihydrochloride POWDER;INTRAVENOUS 209936-001 Sep 14, 2017 DISCN Yes No ⤷  Sign Up ⤷  Sign Up Y Y ⤷  Sign Up
>Applicant >Tradename >Generic Name >Dosage >NDA >Approval Date >TE >Type >RLD >RS >Patent No. >Patent Expiration >Product >Substance >Delist Req. >Patented / Exclusive Use >Submissiondate

Foreign Priority and PCT Information for Patent: 7,511,041

Foriegn Application Priority Data
Foreign Country Foreign Patent Number Foreign Patent Date
02021861Sep 30, 2002
PCT Information
PCT FiledSeptember 18, 2003PCT Application Number:PCT/EP03/10377
PCT Publication Date:April 08, 2004PCT Publication Number: WO2004/029055

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