Understanding the Scope and Claims of United States Patent 9,714,258
Introduction to Patent 9,714,258
United States Patent 9,714,258, titled "Diaryl macrocycles as modulators of protein kinases," is a patent that delves into the development and application of specific chemical compounds. Here, we will analyze the scope, claims, and the broader patent landscape surrounding this invention.
Overview of the Invention
The patent describes certain diaryl macrocyclic compounds, their pharmaceutical compositions, and methods of using these compounds as modulators of protein kinases. Protein kinases are enzymes that play crucial roles in various cellular processes, and their dysregulation is often associated with diseases such as cancer and inflammatory disorders[2].
Scope of the Patent
Chemical Compounds
The patent focuses on a class of diaryl macrocyclic compounds, which are characterized by their specific chemical structures. These compounds include various functional groups such as alkyl, fluoro, ethenopyrazolo, methyl, tetrahydro, and others. The detailed description of these compounds highlights their potential therapeutic applications, particularly in modulating protein kinase activity[2].
Pharmaceutical Compositions
The patent also covers pharmaceutical compositions containing these diaryl macrocyclic compounds. These compositions can include various excipients, formulations, and delivery methods, which are essential for the effective administration of the compounds in a clinical setting.
Methods of Use
The methods of using these compounds are a critical aspect of the patent. It outlines how these diaryl macrocyclic compounds can be used to treat or prevent diseases associated with protein kinase dysregulation. This includes detailed protocols for administration, dosage, and potential combination therapies.
Claims of the Patent
Independent Claims
The patent includes several independent claims that define the scope of the invention. These claims typically cover the specific chemical structures of the diaryl macrocyclic compounds, their pharmaceutical compositions, and the methods of using these compounds. For example, Claim 1 might describe a specific diaryl macrocyclic compound with particular functional groups, while Claim 2 might describe a pharmaceutical composition containing this compound.
Dependent Claims
Dependent claims further narrow down the scope of the independent claims by adding additional limitations or features. For instance, a dependent claim might specify a particular dosage form or a specific method of administration.
Patent Landscape Analysis
Importance of Patent Landscape Analysis
Patent landscape analysis is crucial for understanding the broader technological and competitive landscape surrounding a patent. This analysis involves analyzing vast amounts of patent data to extract valuable legal, business, and technical insights[3].
Key Elements of Patent Landscape Analysis
- Application Number, Filing Date, and Country: These details help identify the patent and its status in different countries.
- Legal Status: This includes whether the patent is alive, pending, lapsed, revoked, or expired.
- Expected Expiry Dates: Knowing when patents are expected to expire is vital for planning and strategy.
- Patent Trends and Market Developments: This includes mergers and acquisitions, in/out-licensing, litigation, and opposition activities.
Tools and Resources
Several tools and resources are available for conducting a thorough patent landscape analysis:
- Patent Public Search: A web-based tool provided by the USPTO that offers enhanced access to prior art[4].
- Global Dossier: A service that provides access to the file histories of related applications from participating IP Offices[4].
- Common Citation Document (CCD): Consolidates prior art cited by all participating offices for the family members of a patent application[4].
Competitive Landscape
Identifying Competitors
The patent landscape analysis helps in identifying competitors who are also working on similar technologies. This can include other pharmaceutical companies or research institutions that have filed patents related to protein kinase modulators.
Market Developments
Understanding market developments such as mergers and acquisitions, licensing agreements, and litigation activities can provide insights into the competitive dynamics. For example, if a competitor has recently acquired a company with a similar patent portfolio, it could indicate a shift in the market strategy.
Legal and Business Implications
Patent Validity and Enforcement
The legal status of the patent, including its validity and any potential challenges or oppositions, is crucial for business strategy. Ensuring that the patent is valid and enforceable is essential for protecting intellectual property rights.
Licensing and Collaboration
The patent landscape analysis can also reveal opportunities for licensing or collaboration. If other companies have complementary patents, there may be opportunities for cross-licensing agreements or joint development projects.
Conclusion
United States Patent 9,714,258 is a significant invention in the field of pharmaceuticals, particularly in the modulation of protein kinases. Understanding the scope and claims of this patent, along with a thorough patent landscape analysis, is essential for navigating the competitive landscape and making informed business decisions.
Key Takeaways
- Specific Chemical Compounds: The patent focuses on diaryl macrocyclic compounds with specific functional groups.
- Pharmaceutical Compositions: The patent covers various pharmaceutical compositions and delivery methods.
- Methods of Use: Detailed methods for using these compounds in treating diseases associated with protein kinase dysregulation.
- Patent Landscape Analysis: Essential for understanding the competitive landscape, market developments, and legal implications.
- Tools and Resources: Utilize tools like Patent Public Search, Global Dossier, and CCD for comprehensive analysis.
FAQs
Q1: What is the main focus of United States Patent 9,714,258?
A1: The main focus is on diaryl macrocyclic compounds as modulators of protein kinases.
Q2: What are the key elements of patent landscape analysis?
A2: Key elements include application number, filing date, country, legal status, expected expiry dates, and market developments.
Q3: How can patent landscape analysis help in business strategy?
A3: It helps in identifying competitors, understanding market developments, and revealing opportunities for licensing or collaboration.
Q4: What tools are available for conducting patent landscape analysis?
A4: Tools include Patent Public Search, Global Dossier, and Common Citation Document (CCD).
Q5: Why is it important to know the legal status of a patent?
A5: Knowing the legal status ensures that the patent is valid and enforceable, protecting intellectual property rights.
Sources
- U.S. Patent and Trademark Office (USPTO) | USAGov
- US9714258B2 - Diaryl macrocycles as modulators of protein kinases - Google Patents
- Navigating Technological Domains with Patent Landscape Analysis - Sagacious Research
- Search for patents - USPTO
